AM404/丙烯酰胺404 产品编号:Asc-095 产品规格:10mg/50mg AM404 Anandamide transport inhibitor Purity: >99%
Biological Description
Competitive and selective anandamide transport inhibitor (IC50 = 1 μM). Active in vivo. Does not activate CB1 receptors or inhibit anandamide hydrolysis but has been shown to activate vanilloid receptors.
Useful References
Beltramo et al (1997) Functional role of high-affinity anandamide transport, as revealed by selective inhibition. Science 277:1094-7 abstract
Zygmunt et al (2000) The anandamide transport inhibitor AM404 activates vanilloid receptors. Eur.J.Pharmacol. 396:39-42 abstract
Bortolato et al (2006) Anxiolytic-like properties of the anandamide transport inhibitor AM404. Neuropsychopharmacology. 2006 31:2652-9. abstract