公告提醒:爱必信所有产品和服务仅用于科学研究,不用于临床应用及其他用途提供产品和服务(也不为任何个人提供产品和服务)! 试剂描述: 产品名称:N-Octadecyl-N'-propyl-sulfamide 产品别名:N-Octadecyl-N'-propylsulfuric diamide CAS号:925891-74-3 英文别名:N-Octadecyl-N'-propylsulfuric diamide 分子量:390.7 分子式:C21H46N2O2S 纯度:≥95% 外观:见爱必信官网 保存方法:Store at -20℃ 描述:Peroxisome proliferator-activated receptors (PPARs) play an essential role in regulating lipid and glucose metabolism. Oleoyl ethanolamide (OEA), a natural ligand for PPARα, has been shown to suppress food intake and reduce weight gain in rats when administered systemically at 10 mg/kg intraperitoneally.1,2 N-Octadecyl-N'-propyl-sulfamide is an analog of OEA with selective binding affinity for PPARα. It is a more potent activator of PPARα, exhibiting an EC50 value of 100 nM, compared to OEA, which exhibits an EC50 value of 120 nM.3,2 At a dose of 1 mg/kg for 8-11 days, N-octadecyl-N'-propyl-sulfamide induces satiety, thereby decreasing food-intake, body weight, and plasma triglyceride concentration in free-feeding Wistar and obese Zucker (fa/fa) rats.3 应用:见爱必信官网 产品信息订购: 产品货号 | 产品名称 | 规格 | 价格 | 大包装及货期 | abs47046243 | N-Octadecyl-N'-propyl-sulfamide | 10mg | 3573 | 立即咨询 | 产品更多信息请进入爱必信网站咨询 |