MEK Inhibitor I

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试剂描述：

产品名称：MEK Inhibitor I

产品别名：MEK Inhibitor I

CAS号：297744-42-4

英文别名：MEK Inhibitor I

分子量：374.46

分子式：C₂₁H₁₈N₄OS

纯度：≥95%

外观：见爱必信官网

保存方法：Store at -20° C

描述：MEK Inhibitor I is a cell-permeable, pyridine-containing, vinylogous cyanamide that has the ability to act as a selective and potent inhibitor of MEK with little activity towards MKK3 and MKK4. The compound displays significant affinity only towards ATP-bound MEK (i.e. noncompetitive with respect to ATP) and the demonstrated inhibition is noncompetitive with respect to ERK. Compared to U0126 in aqueous solutionsMEK Inhibitor I demonstrates superior potency, solubility, and stability. Additionally shown to protect against phorbol ester-mediated ear edema in mice.

应用：A vinylogous cyanamide that has the ability to act as a selective and potent inhibitor of MEK

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