公告提醒:爱必信所有产品和服务仅用于科学研究,不用于临床应用及其他用途提供产品和服务(也不为任何个人提供产品和服务)! 试剂描述: 产品名称:TMB-8 • HCl 产品别名:8-(Diethylamino)octyl 3,4,5-trimethoxybenzoate hydrochloride; 3,4,5-Trimethoxybenzoic acid 8-(diethylamino)octyl ester hydrochloride CAS号:53464-72-5 英文别名:8-(Diethylamino)octyl 3,4,5-trimethoxybenzoate hydrochloride; 3,4,5-Trimethoxybenzoic acid 8-(diethylamino)octyl ester hydrochloride 分子量:431.99 分子式:C22H37NO5•HCl 纯度:≥98% 外观:见爱必信官网 保存方法:Store at 4° C 描述:TMB-8•HCl is a protein kinase C (PKC) inhibitor which also serves as an intracellular Ca2+ antagonist. TMB-8 possesses both Ca2+ channel- and Na+ channel-blocking properties and reduces the membrane K+ conductance. Shown to nonselectively inhibit membrane currents in single isolated guinea pig ventricular cardiomyocytes and to inhibit 5-hydroxytryptamine type 3A (5-HT3A, SR-3A) receptor-mediated currents. TMB-8 inhibits platelet-activating factors (PAF) and PMA-stimulated prostaglandin production in Kupffer cells. Research shows that TMB-8 accumulates at the lipid-water interphase of biologic membranes and therefore interferes with the normal function of many membrane proteins. A useful tool to distinguish dependence on intracellular versus extracellular Ca2+. 应用:A PKC inhibitor and a calcium and sodium channel blocker 产品信息订购: 产品货号 | 产品名称 | 规格 | 价格 | 大包装及货期 | abs42028489 | TMB-8 • HCl | 10mg | 697 | 立即咨询 | 产品更多信息请进入爱必信网站咨询 |