PSB 10,PSB 10 hydrochloride,8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-onemonohydrochloride,591771-91-4

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试剂描述：

产品名称：PSB 10

产品别名：8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride

CAS号：591771-91-4

英文别名：8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride

分子量：435.14

分子式：C₁₆H₁₄Cl₃N₅O•HCl

纯度：见爱必信官网

外观：见爱必信官网

保存方法：Desiccate at 4° C

描述：PSB 10 is a potent and highly selective antagonist for the human Adenosine A3-R, with low affinity for the rat Adenosine A3-R (K_i values are 0.44 and > 17000 nM, respectively). PSB 10 Displays > 3800-fold selectivity over human Adenosine A1-R, Adenosine A2A-R and Adenosine A2B-R (K_i values are 4.1, 3.3 and 30 μM, respectively) and > 1800-fold selectivity over rat Adenosine A1-R and Adenosine A2A-R. This compound acts as an inverse agonist in the [35S]GTPγS binding assay in hA3-CHO cells (IC₅₀ = 4 nM).

应用：A potent and highly selective antagonist for the Adenosine A3-R

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