公告提醒:爱必信所有产品和服务仅用于科学研究,不用于临床应用及其他用途提供产品和服务(也不为任何个人提供产品和服务)! 试剂描述: 产品名称:PDGFR Tyrosine Kinase Inhibitor III 产品别名:4-(6,7-dimethoxyquinazolin-4-yl)-N-(4-phenoxyphenyl)piperazine-1-carboxamide CAS号:205254-94-0 英文别名:4-(6,7-dimethoxyquinazolin-4-yl)-N-(4-phenoxyphenyl)piperazine-1-carboxamide 分子量:485.5 分子式:C27H27N5O4 纯度:见爱必信官网 外观:见爱必信官网 保存方法:Store at 4° C 描述:PDGFR Tyrosine Kinase Inhibitor III is a cell-permeable, potent, selective, and ATP-competitive inhibitor of the PDGFR family of tyrosine kinases (IC50 = 50 nM for PDGFR-α, 80 nM for PDGFR-β, 50 nM for c-Kit, and 230 nM for Flt-3/Flk-2). PDGFR Tyrosine Kinase Inhibitor III inhibits the activities of other kinases only at much higher concentrations (IC50 > 30μM for EGFR, FGFR, Src, PKA, and PKC). Reported to block PDGF-BB-induced proliferation of porcine aorta smooth muscle cells (IC50 = 250 nM). 应用:An ATP-competitive PDGFR inhibitor 产品信息订购: 产品货号 | 产品名称 | 规格 | 价格 | 大包装及货期 | abs42024785 | PDGFR Tyrosine Kinase Inhibitor III | 1mg | 2028 | 立即咨询 | 产品更多信息请进入爱必信网站咨询 |