公告提醒:爱必信所有产品和服务仅用于科学研究,不用于临床应用及其他用途提供产品和服务(也不为任何个人提供产品和服务)! 试剂描述: 产品名称:PAC-1 产品别名:4-(Phenylmethyl)-�1-piperazineacetic Acid� 2-[[2-Hydroxy-3-(2-propen-1-yl)phenyl]methylene]hydrazide; �Procaspase Activating Compound 1 CAS号:315183-21-2 英文别名:4-(Phenylmethyl)-�1-piperazineacetic Acid� 2-[[2-Hydroxy-3-(2-propen-1-yl)phenyl]methylene]hydrazide; �Procaspase Activating Compound 1 分子量:392.49 分子式:C23H28N4O2 纯度:见爱必信官网 外观:见爱必信官网 保存方法:见爱必信官网 描述: PAC-1 is a caspase 3 activator. Caspase activation is a key strategy in cancer therapy. Caspase 3 is a key executioner caspase and direct effector of apoptosis. Hallmark of many cancers is the circumvention of signal in the activation of executioner caspases and loss of apoptotic response. EC50 for caspase 3 activation = 0.33 μM and caspase 7= 4.5 μM. The IC50 for apoptosis induction = 0.92 μM. Elevated caspase 3 level in cancerous cell lines and tissues allows PAC-1 to selectively induce apoptosis in tissues. 应用:见爱必信官网 产品信息订购: 产品货号 | 产品名称 | 规格 | 价格 | 大包装及货期 | abs44127929 | PAC-1 | 25mg | 1750 | 立即咨询 | 产品更多信息请进入爱必信网站咨询 |