公告提醒:爱必信所有产品和服务仅用于科学研究,不用于临床应用及其他用途提供产品和服务(也不为任何个人提供产品和服务)! 试剂描述: 产品名称:Astemizole-d3 产品别名:1-[(4-fluorophenyl)methyl]-N-[1-[2-[4-(trideuteriomethoxy)phenyl]ethyl]piperidin-4-yl]benzimidazol-2-amine CAS号:1189961-39-4 英文别名:1-[(4-fluorophenyl)methyl]-N-[1-[2-[4-(trideuteriomethoxy)phenyl]ethyl]piperidin-4-yl]benzimidazol-2-amine 分子量:461.59 分子式:C28H28D3FN4O 纯度:见爱必信官网 外观:见爱必信官网 保存方法:Store at -20° C 描述:Astemizole-d3 is a labeled form of Astemizole which functions as a non-sedating type histamine H1-receptor anatagonist. Studies suggest that Astemizole-d3 inhibits channels encoded by the gene HERG in Xenopus oocytes via a voltage dependent mechanism. In addition, Astemizole-d3 blocks hEag1 K+ channels which in turn results in inhibiting the expression of cyclins D1 and E. Astemizole-d3 potentiates the anticancer activity of doxorubicin via inhibiting P-glycoprotein pump-efflux activity on human leukemia cells (K-562/DXR) in a dose-related manner. 应用:A labeled histamine H1-receptor anatagonist 产品信息订购: 产品货号 | 产品名称 | 规格 | 价格 | 大包装及货期 | abs42013566 | Astemizole-d3 | 1mg | 4950 | 立即咨询 | 产品更多信息请进入爱必信网站咨询 |