BQ-610,(2R)-2-[[(2R)-2-[[(2S)-2-(azepane-1-carbonylamino)-4-methylpentanoyl]amino]-3-(1-formylindol-3-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoic acid,141595-53-1

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试剂描述：

产品名称：BQ-610

产品别名：Hexahydroazepinocarbonyl-leucyl-tryptophyl(cho)-tryptophan

CAS号：141595-53-1

英文别名：Hexahydroazepinocarbonyl-leucyl-tryptophyl(cho)-tryptophan

分子量：656.7

分子式：C₃₆H₄₄N₆O₆

纯度：≥90%

外观：Powder

保存方法：Store at -20° C

描述：BQ-610 is a highly selective ETAR (ET_A receptor) antagonist (IC₅₀= 20 nM) which attenuates ET-induced reduction in cardiac output. It also inhibits ET-1- and ET-3-induced activation of adenylate cyclase (IC₅₀= 28.2 nM). BQ-610 is 30-fold more potent than BQ-123, in porcine aortic smooth muscle membrane assay.

应用：A highly selective ET_A receptor antagonist

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