公告提醒:爱必信所有产品和服务仅用于科学研究,不用于临床应用及其他用途提供产品和服务(也不为任何个人提供产品和服务)! 试剂描述: 产品名称:Glucagon Receptor Antagonist I 产品别名:N-(3-Cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydro-1-benzothien-2-yl)-2-ethylbutanamide; hGCGR Antagonist CAS号:438618-32-7 英文别名:N-(3-Cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydro-1-benzothien-2-yl)-2-ethylbutanamide; hGCGR Antagonist 分子量:346.5 分子式:C20H30N2OS 纯度:>95% 外观:见爱必信官网 保存方法:Store at 4° C 描述:Glucagon Receptor Antagonist I is a potent and selective cell-permeable thienyl-amide compound that acts as a competitive antagonist of the glucagon receptor. Exhibits binding to hGCGR with high affinity and prevents its interaction with glucagon (IC50 = 181 nM, KDB = 81 nM, and pA2 = 7.1 in membranes prepared from CHO-hGCGR). Also suppresses glucagon-induced glycogenolysis in human primary hepatocytes and in mice (50 mg/kg, ip). 应用:A potent and selective cell-permeable glucagon receptor antagonist 产品信息订购: 产品货号 | 产品名称 | 规格 | 价格 | 大包装及货期 | abs42019039 | Glucagon Receptor Antagonist I | 1mg | 1820 | 立即咨询 | 产品更多信息请进入爱必信网站咨询 |