公告提醒:爱必信所有产品和服务仅用于科学研究,不用于临床应用及其他用途提供产品和服务(也不为任何个人提供产品和服务)! YZ剂描述: 产品名称:Desipramine hydrochloride 产品别名:盐酸去甲咪嗪 英文别名:Desipramine hydrochloride 靶点:5-HT Receptor CAS:58-28-6 纯度:>98% 外观:white to off-white powder 保存方法:store at -20℃ for one year(Powder); in DMSO or others solvent store at 2-4℃ for two weeks, at -20℃ for six months. 描述: Desipramine Hydrochloride a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine. In the central nervous system (CNS), desipramine hydrochloride blocks the re-uptake of neurotransmitters, including norepinephrine and serotonin. This leads to an increase in the amount of these neurotransmitters in the synaptic cleft and prolongs their activities postsynaptically. 溶解性:DMSO : 83.3 mg/mL (275.06 mM; Need ultrasonic and warming) 体外研究: 体内研究:Treatment of rats with Desipramine hydrochloride for 14 days reduces norepinephrine transporter (NET) expression in a dose-dependent manner, as indicated by a reduction of the specific binding of 3H-nisoxetine to the NET in preparations of cerebral cortex (F(3,16)=4.33, p(3,16)=4.34, p. 产品信息订购: 产品货号 | 产品名称 | 规格 | 价格 | 大包装及货期 | abs816997 | Desipramine hydrochloride | 25mg | 550 | 立即咨询 | 产品更多信息请进入爱必信网站咨询 |