公告提醒:爱必信所有产品和服务仅用于科学研究,不用于临床应用及其他用途提供产品和服务(也不为任何个人提供产品和服务)! YZ剂描述: 产品名称:Alosetron (Z)-2-butenedioate 产品别名:(Z)-but-2-enedioic acid,5-methyl-2-[(5-methyl-1H-imidazol-4-yl)methyl]-3,4-dihydropyrido[4,3-b]indol-1-one 英文别名:Alosetron ((Z)-2-butenedioate) 靶点:5-HT Receptor CAS:122852-43-1 纯度:见爱必信官网 外观:见爱必信官网 保存方法:见爱必信官网 描述:Alosetron (Z)-2-butenedioate (GR 68755 (Z)-2-butenedioate) is a Serotonin 5HT3-receptor antagonist that is used in treatment of irritable bowel syndrome.IC50 Value: N/ATarget: 5-HT ReceptorAlosetron has an antagonist action on the 5-HT3 receptors of the enteric nervous system of the gastrointestinal tract. While being a 5-HT3 antagonist like ondansetron, it is not classified or approved as an antiemetic. Since stimulation of 5-HT3 receptors is positively correlated with gastrointestinal motility, alosetron's 5-HT3 antagonism slows the movement of fecal matter through the large intestine, increasing the extent to which water is absorbed, and decreasing the moisture and volume of the remaining waste products. From Wikipedia. 溶解性:10 mM in DMSO 体外研究: 体内研究: 产品信息订购: 产品货号 | 产品名称 | 规格 | 价格 | 大包装及货期 | abs819099 | Alosetron (Z)-2-butenedioate | 10mg | 759 | 立即咨询 | 产品更多信息请进入爱必信网站咨询 |