公告提醒:爱必信所有产品和服务仅用于科学研究,不用于临床应用及其他用途提供产品和服务(也不为任何个人提供产品和服务)! YZ剂描述: 产品名称:Gemcitabine 产品别名:吉西他滨 英文别名:NSC 613327;LY188011 靶点:DNA_RNA Synthesis CAS:95058-81-4 纯度:>98% 外观:白色至浅黄色粉末 保存方法:store at -20℃ for one year(Powder); in DMSO or others solvent store at 2-4℃ for two weeks, at -20℃ for six months. 描述: Gemcitabine is a nucleoside metabolic inhibitor in PANC1(IC50=50 nM), MIAPaCa2(IC50=40 nM), BxPC3(IC50=18 nM) and Capan2 cells(IC50=12 nM). 溶解性:DMSO : 15 mg/mL (56.99 mM) 体外研究: MTS assay demonstrates that Gemcitabine at 15 nM, indole-3-carbinol (I3C) at 50 μM and the combination does not affect hTERT-HPNE cell viability. However, treatment with Gemcitabine at 15 nM, I3C at 50 μM and the combination results in 31%, 19% and 72% cell death of BxPC-3 cells, respectively. 体内研究:Treatment of the LSL-KrasG12D/+; LSL-Trp53R172H; Pdx-1-Cre mice with either Gemcitabine (50 mg/kg, i.p.) or the combination DMAPT/Gemcitabine significantly increased the median survival time by more than 30 days compared to the placebo group (254.5 or 255 days vs. 217.5 days, respectively). Gemcitabine can be administered via endotracheal spray in rats without marked toxicity with a maximum tolerated dose of 4 mg/kg once a week for 9 weeks. The toxicity of Gemcitabine is lower via lung than oral administration at dosages of 2, 4, and 6 mg/kg. 产品信息订购: 产品货号 | 产品名称 | 规格 | 价格 | 大包装及货期 | abs814679 | Gemcitabine | 10mg | 480 | 立即咨询 | 产品更多信息请进入爱必信网站咨询 |