货号:
T4657b
CAS号:
211555-05-4
供应商:
安徽经科生物技术有限公司
数量:
库存数量:2
英文名:
WHI-P97
保质期:
最新包装
保存条件:
见产品外包装
规格:
2mg/5mg/10mg
规格: |
2mg |
产品价格: |
¥798.0 |
规格: |
5mg |
产品价格: |
¥1228.0 |
规格: |
10mg |
产品价格: |
¥1818.0 |
英文名称:WHI-P97
中文名称:4-(3',5'-二溴-4-羟基苯基)氨基-6,7-二甲氧基喹唑啉
CAS:211555-05-4
分子式:C16H13Br2N3O3
分子量:455.1
产品说明:WHI-P97 is a rationally designed potent inhibitor of JAK-3. IC50 value: Target: JAK3 Treatment of mast cells with WHI-P97 inhibited the translocation of 5-lipoxygenase (5-LO) from the nucleoplasm to the nuclear membrane and consequently 5-LO-dependent leukotriene (LT) synthesis after IgE receptor/FcepsilonRI crosslinking by >90% at low micromolar concentrations. WHI-P97 did not directly inhibit the enzymatic activity of 5-LO, but prevented its translocation to the nuclear membrane without affecting the requisite calcium signal.点击 这里 联系客服或咨询更多产品详情!
温馨提示:不可用于临床ZL。