货号:
T3712b
CAS号:
1445993-26-9
供应商:
安徽经科生物技术有限公司
数量:
库存数量:2
英文名:
Mivebresib
保质期:
最新包装
保存条件:
见产品外包装
规格:
2mg/5mg/10mg
规格: |
2mg |
产品价格: |
¥732.0 |
规格: |
5mg |
产品价格: |
¥970.0 |
规格: |
10mg |
产品价格: |
¥1735.0 |
英文名称:Mivebresib
中文名称:米维布塞
CAS:1445993-26-9
分子式:C22H19F2N3O4S
分子量:459.11
产品说明:Mivebresib, also known as ABBV-075, is a potent BET inhibitor (bromodomain (BRD)-containing protein) with potential antineoplastic activity. Upon administration, the bromodomain inhibitor ABBV-075 binds to the acetyl-lysine binding site in the BRD of certain BRD-containing protein(s), thereby preventing the interaction between those proteins and acetylated histones. This disrupts chromatin remodeling, prevents the expression of certain growth-promoting genes, and leads to an inhibition of cell growth in susceptible tumors. Also a potent inhibitor of MYC and the TMPRSS2-ETS fusion proteins.点击 这里 联系客服或咨询更多产品详情!
温馨提示:不可用于临床ZL。