Smartox Biotechnology是WY一家专门生产动物毒液多肽毒素,用于细胞离子通道功能研究的生物医药公司。多肽毒素在生物制药领域具有重要的使用价值。Catalog N° 08CON003ω-CONOTOXIN GVIA / Omega conotoxin GVIASelective blocker of Cav2.2 channel ω-conotoxin GVIA (omega conotoxin GVIA) has been isolated from the venom of the cone Conus geographus. ω-conotoxin GVIA acts at presynaptic membranes. It binds and blocks specifically voltage-dependent N-type Ca2+channels Cav2.2 channel with an ED50 of 68pM.
ω-conotoxin GVIA technical informationAA sequence: H-Cys1-Lys-Ser-Hyp-Gly-Ser-Ser-Cys8-Ser-Hyp-Thr-Ser-Tyr-Asn-Cys15-Cys16-Arg-Ser-Cys19-Asn-Hyp-Tyr-Thr-Lys-Arg-Cys26-Tyr-NH2
Hyp: hydroxyproline
(Disulfide bonds between Cys1-Cys16, Cys8-Cys19 and Cys15-Cys26)
Length (aa): 27
Formula: C120H182N38O43S6
Molecular Weight: 3036.05 Da
Appearance: White lyophilized solid
Solubility: water and saline buffer
CAS number: [106375-28-4]
Source: Synthetic
Purity rate: > 95 %
08CON003-00100 | ω-conotoxin GVIA | 0.1mg |
08CON003-00500 | ω-conotoxin GVIA | 0.5mg |
08CON003-01000 | ω-conotoxin GVIA | 1mg |
温馨提示:不可用于临床ZL。