CAS号:
914471-09-3
数量:
200G
规格:
根据定制需求
产品描述:INCB024360 is a potent IDO1 inhibitor(IC50=10 nM) with desirablepharmaceutical properties, which is poised to start clinical trials incancer patients. IC50 Value: 10 nM [1] Target: IDO1 in vitro: Incellular assays,INCB024360 selectively inhibits human IDO1 with IC(50)values of approximately 10nM, demonstrating little activity againstother related enzymes such as IDO2 or tryptophan 2,3-dioxygenase (TDO)[1]. INCB024360