Ciproxifan hydrochloride,Ciproxifan hydrochloride,1049741-81-2

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产品名称：Ciproxifan hydrochloride

产品别名：Ciproxifan hydrochloride

CAS号：1049741-81-2

英文别名：Ciproxifan hydrochloride

分子量：306.79

分子式：C₁₆H₁₈N₂O₂•HCl

纯度：≥98%

外观：见爱必信官网

保存方法：Desiccate at 4° C

描述：Ciproxifan belongs to a novel chemical series of histamine H3-receptor antagonists. In vitro, it behaved as a competitive antagonist at the H3 autoreceptor controlling 3H histamine release from synaptosomes and displayed similar Ki values (0.5-1.9 nM) at the H3 receptor controlling the electrically-induced contraction of guinea pig ileum or at the brain H3 receptor labeled with 125I-iodoproxyfan. This appears to be an orally bioavailable, extremely selective and potent H3-receptor antagonist whose vigilance- and attention-promoting effects are promising for therapeutic applications in aging disorders.

应用：A novel chemical series of histamine H3-receptor antagonists

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