特别提示:包括neurokininNK1受体YZ剂(Rolapitant)在内,本公司的所有产品仅可用于科研实验,严禁用于临床YL及其他非科研用途!
产品名称:neurokininNK1受体YZ剂(Rolapitant)
英文名称:Rolapitant
产品货号:M01371
产品规格:1mL(10mM)|2mg|5mg|10mg|25mg|50mg|100mg
Rolapitant(SCH619734)是GX选择性具有的neurokininNK1受体YZ剂,Ki值为0.66nM。
注:本品仅可用于科研实验,严禁用于临床YL及其他用途!
CAS号:552292-08-7
别名:SCH619734
纯度:98.01%
分子式:C₂₅H₂₆F₆N₂O₂
分子量:500.48
结构式:
储存条件:-20℃,有效期2年,溶入溶剂后-20℃请尽量在一个月内使用。
除了neurokininNK1受体YZ剂(Rolapitant),SCH619734,我公司还供应以下相关产品:
YT330 出核转运YZ剂(Leptomycin B) 10μg
M00007 NEDD8活化酶YZ剂(MLN4924) 1mL(10mM)|1mg|5mg|10mg|50mg|100mg|200mg
M00384 AktYZ剂(GSK-690693) 1mL(10mM)|5mg|10mg|50mg|100mg
M00560 高度PPARδ激动剂(GW0742) 1mL(10mM)|5mg|10mg|50mg|100mg
M00861 PARPYZ剂(AZD-2461) 1mL(10mM)|2mg|5mg|10mg|50mg|100mg
M01034 GSTP1-1YZ剂(Ezatiostat) 1mL(10mM)|5mg|10mg|50mg|100mg
M01277 乙酰-赖氨酸竞争性蛋白-蛋白相互作用YZ剂(I-CBP112) 1mL(10mM)|1mg|5mg|10mg|50mg|100mg
M01290 泛-RafYZ剂(CCT196969) 1mL(10mM)|5mg|10mg|50mg|100mg
M01670 坏死性凋亡YZ剂(Necrostatin 2 S enantiomer) 1mL(10mM)|1mg|5mg|10mg|50mg
M01707 DprE1YZ剂(PBTZ169) 1mL(10mM)|5mg|10mg|50mg|100mg
M01811 farnesyltransferaseYZ剂(Tipifarnib S enantiomer) 1mL(10mM)|2mg|5mg|10mg|50mg
M02083 FGFRYZ剂(NVP-BGJ398 phosphate) 1mL(10mM)|5mg|10mg
M02633 ERRβ/γ激动剂(GSK-4716) 1mL(10mM)|10mg|50mg|100mg
M02728 LXR激动剂(GW3965 hydrochloride) 1mL(10mM)|5mg|10mg|50mg|100mg
M02733 低氧诱导因子脯氨酰羟化酶YZ剂(Daprodustat) 2mg|5mg|10mg|50mg|100mg
M03421 雌激素受体激动剂(Dienestrol) 1mL(10mM)
M03552 二氮杂双*辛烷YZ剂(Relebactam) 1mL(10mM)|1mg|5mg|10mg|25mg|50mg
M03639 hedgehogYZ剂(Mebendazole) 1mL(10mM)|1g
M04246 HCVRNA复制YZ剂(Sofosbuvir impurity H) 1mL(10mM)|1mg|5mg
M04341 NF-κBYZ剂(BAY 11-7082) 1mL(10mM)|5mg|10mg|50mg|100mg
M04561 p38α MAPKYZ剂(BMS-582949 hydrochloride) 1mL(10mM)|1mg|5mg|10mg|25mg|50mg|100mg
M04664 BCL6YZ剂(FX1) 1mL(10mM)|5mg|10mg|25mg|50mg|100mg|200mg
M04710 前列腺素合成YZ剂(Suprofen) 1mL(10mM)|10mg|50mg|100mg
M04881 环氧化酶YZ剂(Ampiroxicam) 1mL(10mM)|10mg|50mg
M05320 XOYZ剂(Febuxostat) 1mL(10mM)|10mg|50mg|100mg
M05797 LRRK2YZ剂(PF-06447475) 1mL(10mM)|5mg|10mg
M06006 TASK-1/TASK-3和TASK-1/TASK-3异二聚体通道YZ剂 1mL(10mM)|50mg|100mg
M06314 组胺H3受体YZ剂 1mL(10mM)|100mg|1g|5g|10g
M06433 单胺氧化酶MAO-AYZ剂(Minaprine) 1mL(10mM)|100mg
M06511 高亲和性A3腺苷受体激动剂(AB-MECA) 1mL(10mM)|1mg|5mg
温馨提示:不可用于临床ZL。