DiscoveryProbe™ Tyrosine Kinase Inhibitor Library_详细资料

产品信息

规格： 100uL/well(10 mM solution)///250uL/well(10 mM solution)///5mg/well

270个酪氨酸激酶YZ剂的独特集合，用于高通量筛选（HTS）和高含量筛选（HCS）

规格单价

100uL/well(10 mM solution) ￥42,200.00

250uL/well(10 mM solution) ￥75,300.00

5mg/well ￥98,400.00

Featured Products of the Library

Catalog No. Product Name Summary Targets CAS Number Smiles

A1389 WZ4002 Mutant-selective EGFR inhibitor(L858R,T790M), irreversible and potent EGFR 1213269-23-8 CN1CCN(CC1)C2=CC(=C(C=C2)NC3=NC=C(C(=N3)OC4=CC=CC(=C4)NC(=O)C=C)Cl)OC

A2838 OSI-930 Inhibitor of Kit, KDR, Flt, CSF-1R, c-Raf and Lck c-Kit 728033-96-3 C1=CC=C2C(=C1)C(=CC=N2)CNC3=C(SC=C3)C(=O)NC4=CC=C(C=C4)OC(F)(F)F

A3014 BGJ398 FGFR inhibitor ,potent and selective FGFR 872511-34-7 CCN1CCN(CC1)C2=CC=C(C=C2)NC3=CC(=NC=N3)N(C)C(=O)NC4=C(C(=CC(=C4Cl)OC)OC)Cl

A5092 JNJ-38877605 C-Met inhibitor,ATP-competitive c-MET 943540-75-8 CN1C=C(C=N1)C2=NN3C(=NN=C3C(C4=CC5=C(C=C4)N=CC=C5)(F)F)C=C2

A8324 LDN-193189 ALK inhibitor,potent and selective SMAD 1062368-24-4 C1CN(CCN1)C2=CC=C(C=C2)C3=CN4C(=C(C=N4)C5=CC=NC6=CC=CC=C56)N=C3

A8329 R428 Selective Axl inhibitor Axl 1037624-75-1 C1CCN(C1)C2CCC3=C(CC2)C=C(C=C3)NC4=NN(C(=N4)N)C5=NN=C6C(=C5)CCCC7=CC=CC=C76

A8528 TAK-285 HER2/EGFR(HER1) inhibitor HER2 871026-44-7 CC(C)(CC(=O)NCCN1C=CC2=C1C(=NC=N2)NC3=CC(=C(C=C3)OC4=CC=CC(=C4)C(F)(F)F)Cl)O

A8696 FIIN-2 Irreversible inhibitor of FGFR EGFR 1633044-56-0 O=C(C=C)NC1=CC=C(CN2C(N(C3=CC(OC)=CC(OC)=C3)CC4=CN=C(NC5=CC=C(N6CCN(C)CC6)C=C5)N=C42)=O)C=C1

Download the Tyrosine-Kinase-Inhibitor-Library - XLSX Download the Tyrosine-Kinase-Inhibitor-Library - SDF

Advantages

Available in stock with overnight delivery and free shipping over $500

Cost-effective and competitive price to save your findings

Potent, selective and cell-permeable in inhibiting or activating target molecules

Diverse in chemical structure and route of administration (oral/i.m/i.v injection etc.)

Detailed files describing potency, selectivity and applications etc.

Supported by published data from top peer-reviewed journals

Guaranteed high quality with NMR and HPLC validation

Storage and Shipping Information

Form Pre-dissolved DMSO solutions Stability -20°C: 12 months
-80°C: 24 months

Packaging 96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode.

General tips For obtaining a higher solubility , please warm the tube at 37°C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months.

Shipping Condition Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request

温馨提示：不可用于临床ZL。

规格	单价
100uL/well(10 mM solution)	￥42,200.00
250uL/well(10 mM solution)	￥75,300.00
5mg/well	￥98,400.00

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Catalog No.	Product Name	Summary	Targets	CAS Number	Smiles
A1389	WZ4002	Mutant-selective EGFR inhibitor(L858R,T790M), irreversible and potent	EGFR	1213269-23-8	CN1CCN(CC1)C2=CC(=C(C=C2)NC3=NC=C(C(=N3)OC4=CC=CC(=C4)NC(=O)C=C)Cl)OC
A2838	OSI-930	Inhibitor of Kit, KDR, Flt, CSF-1R, c-Raf and Lck	c-Kit	728033-96-3	C1=CC=C2C(=C1)C(=CC=N2)CNC3=C(SC=C3)C(=O)NC4=CC=C(C=C4)OC(F)(F)F
A3014	BGJ398	FGFR inhibitor ,potent and selective	FGFR	872511-34-7	CCN1CCN(CC1)C2=CC=C(C=C2)NC3=CC(=NC=N3)N(C)C(=O)NC4=C(C(=CC(=C4Cl)OC)OC)Cl
A5092	JNJ-38877605	C-Met inhibitor,ATP-competitive	c-MET	943540-75-8	CN1C=C(C=N1)C2=NN3C(=NN=C3C(C4=CC5=C(C=C4)N=CC=C5)(F)F)C=C2
A8324	LDN-193189	ALK inhibitor,potent and selective	SMAD	1062368-24-4	C1CN(CCN1)C2=CC=C(C=C2)C3=CN4C(=C(C=N4)C5=CC=NC6=CC=CC=C56)N=C3
A8329	R428	Selective Axl inhibitor	Axl	1037624-75-1	C1CCN(C1)C2CCC3=C(CC2)C=C(C=C3)NC4=NN(C(=N4)N)C5=NN=C6C(=C5)CCCC7=CC=CC=C76
A8528	TAK-285	HER2/EGFR(HER1) inhibitor	HER2	871026-44-7	CC(C)(CC(=O)NCCN1C=CC2=C1C(=NC=N2)NC3=CC(=C(C=C3)OC4=CC=CC(=C4)C(F)(F)F)Cl)O
A8696	FIIN-2	Irreversible inhibitor of FGFR	EGFR	1633044-56-0	O=C(C=C)NC1=CC=C(CN2C(N(C3=CC(OC)=CC(OC)=C3)CC4=CN=C(NC5=CC=C(N6CCN(C)CC6)C=C5)N=C42)=O)C=C1
Download the Tyrosine-Kinase-Inhibitor-Library - XLSX Download the Tyrosine-Kinase-Inhibitor-Library - SDF

Form	Pre-dissolved DMSO solutions	Stability	-20°C: 12 months -80°C: 24 months
Packaging	96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode.
General tips	For obtaining a higher solubility , please warm the tube at 37°C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months.
Shipping Condition	Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request